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Conference Materials

The Conference Program can be downloaded here (link).

The Book of Abstracts can be downloaded here (link).
 
 

8th International Conference “CHEMISTRY OF NITROGEN CONTAINING HETEROCYCLES” in memoriam of Prof. Valeriy Orlov (12th - 16th November, 2018, Kharkiv, Ukraine)

 
Types of reports
PL – plenary lecture (60 min) O – oral report (20 min) INV – invited lecture (30 min) S – short talk (15 min)
 
 
  November 12
V.N. Karazin Kharkov National University
Svobody sq. 4 , Main Building, the 2nd floor, Assembly Hall, reception
Assembly Hall
9:00-13:00
Registration
Assembly Hall
13:00-14:00
Opening ceremony
Assembly Hall
14:00-14:30
Prof. Andrey Doroshenko
V.N.Karazin Kharkov National University Introductory lecture in memoriam of Prof. Valeriy Orlov
14:30-15:30 PL-1
Prof. Erik Van der Eycken
University of Leuven
Synthesis of small complex heterocycles
15:30-15:45 Coffee-break
Assembly Hall Chairman
15:45-16:45 PL-2
Prof. Dmytro Volochnyuk
Enamine Ltd
MedChem-relevant building blocks: from definitions and criteria to part of industry
16:45-17:15 INV-1
Prof. Victoria Lipson
State Institution “V.Ya. Danilevsky Institute for Endocrine Pathology Problems” of the NAMS of Ukraine
Glyoxals, Aminoazoles and CH-Acids in Diversity-oriented Synthesis of Azoloazines
17:15-17:35 O-1
Dr. Maksim Kolosov
V.N.Karazin Kharkov National University
Light” 5-methyl-4,7-dihydroazolo[1,5-a]pyrimidines and related 3,4-dihydropyrimidin-2(1H)-ones
17:35-17:55 O-2
Dr. Esma Abdurakhmanova
Institute of Bioorganic Chemistry and Petrochemistry NAS Ukraine
New phosphonopeptidomimetics: synthesis and properties
17:55-18:30 Free-time
   
   
18:30-20:00

Welcome party

 

  November 13
SSI "Institute for Single Crystals" NAS of Ukraine
Nauky ave. 60, the 5th floor
Large Hall Chairman
9:00-10:00 PL-3
Prof. Alexander Dömling
University of Groningen, Groningen Research Institute of Pharmacy
MCR-chemistry: From automated nano synthesis to novel bioactive scaffolds to natural product synthesis
10:00-10:30 INV-2
Dr. Philippe Gros
Universite de Lorraine/CNRS
Design of new pyridyl N-heterocyclic ligands and corresponding iron complexes: Application to light harvesting and electron-transfer
10:30-10:50 O-3
Dr. Tetiana Pavlovska
SSI "Institute for Single Crystals" NAS of Ukraine
Domino reactions of 2-amino-4-arylimidazoles with carbonyl and methylene active compounds
10:50-11:05 Coffee-break
Large Hall Chairman
 11:05-11:35
INV-3
Dr. Andrii Monastyrskyi
The Scripps Research Institute
Development of dual casein kinase 1δ/1ε inhibitors for treatment of breast cancer
11:35-11:55 O-4
Dr. Oleksandr Kozachenko
Institute of Bioorganic Chemistry and Petrochemistry NAS Ukraine
Syntheses of new azolopyrimidines on the basis of 2 acylamino-3,3-dichloroacrylonitriles
11:55-12:25
O-5
Prof. Victor Markov
Ukrainian State University of Chemical Technology
New examples of rearrangement of heminal oxazines under Vilsmeier-Haack reagent
12:25-12:40 Coffee-break
12:40-13:40 PL-4
Prof. Thomas Müller
Heinrich Heine University Düsseldorf
Diversity-oriented synthesis of aggregation-induced emissive Nitrogen heterocycles
13:40-14:00 O-6
Ms. Alisa Morozova
SSI "Institute for Single Crystals" NAS of Ukraine
Chemical behavior of selected aminoazoles in reactions with pyruvic acids
14:00-15:00 Lunch
Large Hall Chairman
15:00-16:00 PL-5
Prof. Victor Kartsev
InterBioScreen Ltd
Targeted synthesis of natural compound analogs. reactions and rearrangements
16:00-16:20
O-7
Dr. Sergey Ryabukhin
Enamine Ltd
Synthesis of MedChem-relevant gem-difluorocycloalkane building blocks
16:20-16:40 O-8
Dr. Iryna Omelchenko
SSI "Institute for Single Crystals" NAS of Ukraine
Interplay between stacking, C–H…π and C–H…N interactions in the crystals of ortho-substituted 1,10-phenantrolines with aromatic substituents
16:40-16:55 Coffee-break
17:00-18:30 Seminar “Reaxys – the database for Science and Education”
18:30-20:30 Poster session 1-72
Banquet Hall, the 2th floor

 

  November 14
SSI "Institute for Single Crystals" NAS of Ukraine
Nauky ave. 60, the 5th floor
Small Hall
9:00-18:30
Workshop in specific topic “Chemistry for Pharmacy” in russian
Small Hall, the 5th floor
Large Hall Chairman
9:00-10:00
PL-6
Prof. Igor Komarov
Enamine Ltd
(Spiro)heterocycle-containing Peptidomimetics with Photocontrolled Biological Activity
10:00-10:20
O-9
Dr. Vitalii Palchykov
Oles Honchar Dnipro National University
Oxazaheterocycles from epoxy derivatives
10:20-10:40
O-10
Dr. Anton Tverdokhlebov
Enamine Ltd
Synthesis of 2-azolyl-2,2-difluoroethylamines
10:40-11:00
O-11
Dr. Dmytro Sysoiev
University of Konstanz
Photochromism of molecular wires tuned with heterocyclic scaffolds
10:00-11:15
Coffee-break
Large Hall Chairman
11:15-11:45
INV-4
Prof. Andrea Basso
Università di Genova
Synthesis of Nitrogen-containing heterocycles via elaboration of photoinduced multicomponent adducts
11:45-12:05 O-12
Dr. Maryna Kachaeva
Institute of Bioorganic Chemistry and Petrochemistry NAS Ukraine
Anticancer activity of new 1,3-oxazole derivatives: in silico and in vitro
12:05-12:25 O-13
Dr. Mikhailo Slivka
Uzhhorod National University
Production of condensed triazoles via electrophilic heterocyclization
12:25-12:40
Coffee-break
12:40-13:10
INV-5
Prof. Radek Cibulka
University of Chemistry and Technology
Flavins – not only cofactors but also efficient photocatalysts
13:10-13:25 S-1
Mr. Ihor Pokotylo
Ukrainian State University of Chemical Technology
Synthesis of 4H-1,3,5-Oxadiazine Derivatives Based on N-(2,2,2-Trichloro-1-hydroxyethyl)carboxamides
13:25-14:25 Lunch, Banquet Hall, the 2th floor
Large Hall Chairman
14:30-15:00 INV-6
Prof. Zoia Voitenko
Kiev National University Taras Shevchenko
Heterocyclic compounds in cycloaddition reactions as an inexhaustible source of ideas and products for medical chemistry and sustainable development
15:00-15:20 O-14
Dr. Nikolay Semenishyn
A.V. Bogatsky Physico-Chemical Institute of the NAS of Ukraine
Polytopic macrocyclic tetrapyrroles and their lanthanide derivatives
  S-2
Mr. Oleksii Kolomoitsev
V. N. Karazin Kharkiv National University
Photoreactive fused azyridinylpiperazines
15:35-15:50 Coffee-break
  Chairman
15:50-16:20
INV-7
Dr. Nazariy Pokhodylo
Ivan Franko National University of Lviv
The unpredicted courses and unexpected products in the reaction of azides with alkynes (CuAAC) or methylene ketones
16:20-16:35
S-3
Ms. Galyna Grygoriv
National University of Pharmacy
1,2-Benzoxathiin-4(3H)-one 2,2-dioxide as new enolnucleophile in construction of 2-amino-4H-pyran core
16:35-16:50 Coffee-break
16:50-17:10 O-15
Dr. Irina Konovalova
SSI "Institute for Single Crystals" NAS of Ukraine
Using of precision X-ray diffraction studies for the analysis of reactivity and weak intermolecular interactions in 3,4-diamino-1,2,4-triazole and its 5-methyl derivative
17:10-17:30 O-16
Dr. Lidiya Petrushova
National University of Pharmacy
The study of bromination mechanism and analgesic activity of methyl 1-allyl-4-hydroxy- 2,2-dioxo-1H-2λ6,1- benzothiazine-3-carboxylate
17:30-17:50 O-17
Dr. Muhammad Naveed Umar
University of Malakand
Synthesis of chiral Thioureas in water in the presence of sun Light: Precursors for Nitrogen Heterocyclic compounds
17:50-18:05 Ms. Mariia Vodolazhenko
SSI "Institute for Single Crystals" NAS of Ukraine
Directions of one-pot interaction between cyclic and acyclic α-carbonyl CH-acids, DMFDMA and active methylene nitriles in aqueous medium
18:05-18:15 Dr. Marina Teus
Chief-Editor of Journal "Chemistry of Heterocyclic Compounds"
Latvian Institute of Organic Synthesis
18:15-19:00
Free time
19:00-22:00 Banquet
Banquet Hall, the 2th floor
Chairman

 

  November 15
National University of Pharmacy
Valentynivska str. 4
10:00-10:20 Welcoming notes
  Chairman
10:20-10:50 INV-8
Prof. Wim Dehaen
KU Leuven
New efficient methods for the synthesis of 1,2,3-triazoles
10:50-11:10
O-18
Dr. Victor Shtamburg
Ukrainian State University of Chemical Technology
Arylglyoxals as key precursors for the synthesis of aryl(indol-3-yl)benzoins, aryl(fur-2-yl)benzoins, 5-arylthiohydantoins, N-hydroxyhydantoins and N-alkoxyhydantoins
11:10-11:30
O-19
Dr. Hanna Yeromina
National University of Pharmacy
Design of new biologically active substances based on N-(2-hydroxyethyl)-N'-phenylthiourea
11:30-11:45
Coffee-break
  Chairman
11:45-12:15
INV-9
Prof. Thierry Ollevier
Université Laval
New developments using chiral bipyridine diol metal complexes for asymmetric catalysis
12:15-12:35
O-20
Dr. Nikolay Gorobets
SSI "Institute for Single Crystals" NAS of Ukraine
Rapid formation of chemical complexity via a modified Biginelli reaction using 3-amino-1,2,4-triazoles as the urea component
12:35-12:55 O-21
Dr. Kirill Petko
Institute of Organic Chemistry of NAS of Ukraine
The simplest azoles N-difluoromethylation: features and surprises
12:55-13:10
Coffee-break
  Chairman
13:10-13:30 O-22
Prof. Roman Lesyk
Danylo Halytsky Lviv National Medical University
4-Thiazolidinones: medicinal chemistry aspects
13:30-13:50 O-23
Dr. Tetiana Shvydenko
Institute of Organic Chemistry, NAS of Ukraine
Synthesis and biological activity of ellipticine derivatives
13:50-14:10 O-24
Dr. Sergiy Vlasov
National University of Pharmacy
Development of the novel NSAIDs with the core of 5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
14:10-14:40 Closing Ceremony
14:40-16:40 Lunch
17:00-20:00 Sightseeing interactive tour of Kharkiv

 

08:30-18:00 November 16
Interactive trip to Ukrainian Radio Telescope UTR-2